Development and pharmacological evaluation of a new chemical series of potent pan-ERR agonists, identification of SLU-PP-915

Carissa S. Hampton, Sadichha Sitaula, Cyrielle Billon, Keith Haynes, Amer Avdagic, Udayanga Wanninayake, Christiana M. Adeyemi, Arindam Chatterjee, Kristine Griffett, Subhashis Banerjee, Sheryl L. Burris, Emmalie Schoepke, Terri Boehm, Alex Bess, Ian Mitchelle S. de Vera, Thomas P. Burris, John K. Walker

Research output: Contribution to journalArticlepeer-review

Original languageEnglish
Article number115582
JournalEuropean Journal of Medicinal Chemistry
Volume258
DOIs
StatePublished - Oct 5 2023

ASJC Scopus Subject Areas

  • Pharmacology
  • Drug Discovery
  • Organic Chemistry

Keywords

  • 2 5-disubstituted thiophenes
  • Boronic acid
  • Estrogen-related receptor
  • Nuclear receptor
  • Pan-agonist

Cite this