Development and pharmacological evaluation of a new chemical series of potent pan-ERR agonists, identification of SLU-PP-915

  • Carissa S. Hampton
  • , Sadichha Sitaula
  • , Cyrielle Billon
  • , Keith Haynes
  • , Amer Avdagic
  • , Udayanga Wanninayake
  • , Christiana M. Adeyemi
  • , Arindam Chatterjee
  • , Kristine Griffett
  • , Subhashis Banerjee
  • , Sheryl L. Burris
  • , Emmalie Schoepke
  • , Terri Boehm
  • , Alex Bess
  • , Ian Mitchelle S. de Vera
  • , Thomas P. Burris
  • , John K. Walker

Research output: Contribution to journalArticlepeer-review

Original languageEnglish
Article number115582
JournalEuropean Journal of Medicinal Chemistry
Volume258
DOIs
StatePublished - Oct 5 2023

ASJC Scopus Subject Areas

  • Pharmacology
  • Drug Discovery
  • Organic Chemistry

Keywords

  • 2 5-disubstituted thiophenes
  • Boronic acid
  • Estrogen-related receptor
  • Nuclear receptor
  • Pan-agonist

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