Modulation of estrogen-related receptors subtype selectivity: Conversion of an ERRβ/γ selective agonist to ERRα/β/γ pan agonists

  • Mohamed Shahien
  • , Mohamed Elagawany
  • , Sadichha Sitaula
  • , Shaimaa S. Goher
  • , Sheryl L. Burris
  • , Ryan Sanders
  • , Amer Avdagic
  • , Cyrielle Billon
  • , Lamees Hegazy
  • , Thomas P. Burris
  • , Bahaa Elgendy

Research output: Contribution to journalArticlepeer-review

Original languageEnglish
Article number104079
JournalBioorganic Chemistry
Volume102
DOIs
StatePublished - Sep 2020

ASJC Scopus Subject Areas

  • Biochemistry
  • Molecular Biology
  • Drug Discovery
  • Organic Chemistry

Keywords

  • Estrogen-Related Receptors
  • Molecular Modeling
  • N-Acyl Hydrazones
  • Pan Agonists

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